VEXAS, Vacuoles, E1 enzyme, X-linked, Autoinflammatory, Somatic; mg, milligrams; GC, Glucocorticoid; EOW, End of Week
aPatients who are stable on GC doses of 10-14 mg daily in addition to another non-GC anti-inflammatory therapy at Screening who have a previously documented VEXAS flare on GC monotherapy at a dose of ≥10 mg may be eligible, provided their GC dose is escalated to 15-45mg daily after washout.
bTime periods for washout are variable based on type of non-GC anti-inflammatory therapy
*Anti-CD20 agents (e.g., rituximab): 180 days, Anti-IL-23 agents (e.g., ustekinumab): 90 days, Anti-TNFα except for etanercept (e.g., infliximab): 60 days, Canakinumab: 60 days, Intravenous anti-IL-6 agents (e.g., tocilizumab): 42 days, Subcutaneous anti-IL-6 agents: 28 days, Anti-IL-17 agents (e.g., secukinumab): 28 days, Anti-integrins (e.g., vedolizumab): 60 days, Intravenous immunoglobulin: 28 days, Danazol, immunomodulatory imide drugs (ImiDs), luspatercept, or thrombopoietin receptor agonists: 28 days, Cytotoxic chemotherapy: 28 days, Etanercept: 21 days, Oral Janus kinase (JAK) inhibitors: 14 days, Anti-IL-1 agents except for canakinumab: 14 days, Any other non-GC anti-inflammatory therapy (e.g., mycophenolate, azathioprine, cyclosporine, sulfasalazine, methotrexate): 14 days
Pacritinib (commercially known as VONJO®) was approved by U.S. Food and Drug Administration (FDA) on February 28, 2022 for the treatment of adults with myelofibrosis with a platelet count below 50 x 109/L, and has since been marketed in the US under the brand name VONJO®. This indication is approved under accelerated approval based on spleen volume reduction. Continued approval for this indication may be contingent upon verification and description of clinical benefit in a confirmatory trial(s).